Structure Activity Relationships for Intracellular Loop 2 of the 5HT1A Serotonin Receptor
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چکیده
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منابع مشابه
Intracellular Loop 2 Peptides of the Human 5HT1a Receptor are Differential Activators of Gi
Peptide mimics of intracellular loop 2 (ic2) of the human 5HT1a receptor have been studied with respect to their ability to inhibit agonist binding via interference with receptor-G-protein coupling. These peptides give shallow concentration-effect relationships. Additionally, these peptides have been studied with respect to their ability to trigger the signal transduction system of this Gi-coup...
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